SCHEMBL7705975

SCHEMBL7705975

Nc1cc(N2CCc3c([nH]c4ccccc34)C2)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.48
DHFR P00374 1/20 0.42
KDM4E B2RXH2 1/20 0.41
TRPV1 Q8NER1 3/20 0.41
CDK4 P11802 7/20 0.40
CCND1 P24385 7/20 0.40
FAAH O00519 1/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
GABRA4 P48169 1/20 0.39
GABRE P78334 1/20 0.39
GABRA6 Q16445 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703248 0.86 ADORA2A (0.46) GBA1DHFRKDM4E
SCHEMBL7709059 0.75 SMN1; SMN2 (0.45) KDM4EMEN1KMT2AGAA
SCHEMBL7705992 0.74 HPGD (0.45) KDM4EMEN1KMT2AGAA
SCHEMBL7436334 0.72 HTT (0.50) KDM4EMEN1KMT2AGAA
SCHEMBL21588453 0.69 KDM4E (0.51) DHFRKDM4ETRPV1SIGMAR1MEN1
SCHEMBL21588421 0.69 DHFR (0.53) GBA1DHFRKDM4ETRPV1FAAH
SCHEMBL6867881 0.68 ADORA2A (0.63) CDK4CCND1
SCHEMBL6262143 0.68 KDM4E (0.49) GBA1DHFRKDM4ETRPV1SIGMAR1
SCHEMBL21588327 0.66 KDM4E (0.56) KDM4ETRPV1SIGMAR1MEN1KMT2A
SCHEMBL7423524 0.66 ALDH1A1 (0.53) KDM4EMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed