SCHEMBL7703705

SCHEMBL7703705

C=CCON1C(=O)c2ccc(Cl)c3c(N4CCCC4)cc(NC(C)=O)c(c23)C1=O

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 6/20 0.34
MEN1 O00255 4/20 0.34
TDP1 Q9NUW8 2/20 0.34
CRHBP P24387 1/20 0.34
MAPK1 P28482 1/20 0.34
CRHR2 Q13324 1/20 0.34
ATAD2 Q6PL18 1/20 0.33
CECR2 Q9BXF3 1/20 0.33
KCNQ2 O43526 2/20 0.33
MAPT P10636 3/20 0.33
LMNA P02545 1/20 0.33
KDM4E B2RXH2 1/20 0.32
RECQL P46063 1/20 0.32
HTR2C P28335 1/20 0.32
POLB P06746 2/20 0.31
TP53 P04637 1/20 0.31
BRD4 O60885 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703708 0.85 ALDH1A1 (0.44) ALDH1A1KMT2AMEN1TDP1CRHBP
SCHEMBL7709358 0.81 MAPT (0.40) ALDH1A1KMT2AMEN1TDP1ATAD2
SCHEMBL7706801 0.73 ALDH1A1 (0.55) ALDH1A1KMT2AMEN1TDP1MAPT
SCHEMBL7706701 0.70 MEN1 (0.47) ALDH1A1KMT2AMEN1TDP1CRHBP
SCHEMBL8578190 0.69 TDP1 (0.44) KMT2AMEN1TDP1MAPK1MAPT
SCHEMBL7709710 0.68 MEN1 (0.47) ALDH1A1KMT2AMEN1TDP1CRHBP
SCHEMBL7706698 0.64 MAPT (0.44) ALDH1A1KMT2AMEN1TDP1MAPK1
SCHEMBL7706710 0.62 TYMS (0.45) ALDH1A1KMT2AMEN1MAPTLMNA
SCHEMBL7706707 0.58 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1TDP1MAPK1
SCHEMBL10776759 0.58 CHRM1 (0.49) ALDH1A1KMT2AMEN1TDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed