SCHEMBL7703797

SCHEMBL7703797

CC(=O)Nc1cc2c3c(cccc3c1N1CCCC1)C(=O)N(OC(C)(C)C)C2=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
BRD4 O60885 2/20 0.39
MEN1 O00255 10/20 0.39
KMT2A Q03164 10/20 0.39
USP2 O75604 5/20 0.39
BLM P54132 1/20 0.39
HTT P42858 4/20 0.36
LMNA P02545 4/20 0.36
XBP1 P17861 1/20 0.36
HIF1A Q16665 1/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
TLR9 Q9NR96 2/20 0.36
TNNI3 P19429 1/20 0.36
TNNT2 P45379 1/20 0.36
TNNC1 P63316 1/20 0.36
MAPT P10636 5/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7706721 0.85 HTT (0.50) ALDH1A1KDM4EGAABRD4MEN1
SCHEMBL7706744 0.82 ALDH1A1 (0.46) ALDH1A1KDM4EGAABRD4MEN1
SCHEMBL7709480 0.78 ALDH1A1 (0.62) ALDH1A1GAAMEN1KMT2AHTT
SCHEMBL7703741 0.69 MDM4 (0.39) ALDH1A1KDM4EGAABRD4KMT2A
SCHEMBL7709632 0.68 CYP1B1 (0.58) ALDH1A1KDM4EMEN1KMT2ALMNA
SCHEMBL7703735 0.67 KDM4E (0.44) ALDH1A1KDM4EMEN1KMT2AUSP2
SCHEMBL7709992 0.67 BRD4 (0.45) ALDH1A1BRD4MEN1KMT2AUSP2
SCHEMBL7709561 0.67 BRD1 (0.40) ALDH1A1KDM4EBRD4KMT2ALMNA
SCHEMBL7712199 0.66 KMT2A (0.64) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL5964469 0.66 ALDH1A1 (0.71) ALDH1A1KDM4EGAABRD4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed