SCHEMBL7703836

SCHEMBL7703836

O=C(O)N[C@H]1CCN(c2c(Br)cc3c4c(cccc24)C(=O)N(OCc2ccccc2)C3=O)C1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSK P43235 1/20 0.35
CYP1B1 Q16678 3/20 0.35
MTNR1A P48039 4/20 0.34
MTNR1B P49286 4/20 0.34
CREBBP Q92793 2/20 0.34
PPARG P37231 1/20 0.34
BACE1 P56817 1/20 0.33
ME3 Q16798 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703898 0.88 CTSL (0.39) DRD2DRD4DRD3CTSLCTSB
SCHEMBL7703947 0.82 MEN1 (0.39) CYP1B1
SCHEMBL7706731 0.82 CYP1B1 (0.45) CYP1B1
SCHEMBL7706752 0.81 CYP1B1 (0.44) CYP1B1
SCHEMBL7703698 0.79 CYP1B1 (0.41) SIGMAR1CYP1B1
SCHEMBL7703741 0.73 MDM4 (0.39) MTNR1AMTNR1B
SCHEMBL7703721 0.73 CYP1B1 (0.46) CYP1B1
SCHEMBL7709722 0.71 LMNA (0.36) CTSLCTSBCTSKMTNR1AMTNR1B
SCHEMBL7712197 0.71 CYP1B1 (0.65) CYP1B1
SCHEMBL7712257 0.70 MEN1 (0.46) CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed