SCHEMBL7704394

SCHEMBL7704394

COc1cc(NC(=O)OC(C)(C)C)c(NC(=O)CC(=O)c2ccccc2-n2ccnn2)cc1-c1ccccc1F

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
KMT2A Q03164 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
TSHR P16473 1/20 0.36
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
IDO1 P14902 1/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462988 0.87 CYP17A1 (0.37) IDO1
SCHEMBL7139910 0.80 CYP3A4 (0.34) ALDH1A1TSHR
SCHEMBL7139681 0.79 TSHR (0.36) KMT2ATSHRMEN1
SCHEMBL6165283 0.78 NOTUM (0.34) ALDH1A1TSHRTP53
SCHEMBL6607768 0.78 RXFP1 (0.36) LMNAPOLBIDO1
SCHEMBL7138174 0.78 EGLN2 (0.37) ALDH1A1LMNAKMT2ANPSR1TSHR
SCHEMBL7139741 0.77 TUBB4A (0.38) ALDH1A1LMNAKMT2ATSHRTP53
SCHEMBL7143167 0.76 ABL1 (0.41) ALDH1A1KMT2AMEN1CYP1A2CYP2C19
SCHEMBL7141959 0.76 ALDH1A1 (0.41) ALDH1A1LMNAKMT2ATSHRTP53
SCHEMBL7140010 0.76 MEN1 (0.36) ALDH1A1LMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed