SCHEMBL7704458

SCHEMBL7704458

COc1ccc(-c2cccc3ccccc23)c(Oc2ccccc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.48
CYP11B2 P19099 2/20 0.48
CYP17A1 P05093 1/20 0.48
HDAC8 Q9BY41 1/20 0.46
LTA4H P09960 1/20 0.46
CYP1A2 P05177 3/20 0.45
CYP2A6 P11509 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2B6 P20813 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP1A1 P04798 1/20 0.45
CYP2E1 P05181 1/20 0.45
CYP2C8 P10632 1/20 0.45
CYP4B1 P13584 1/20 0.45
CYP3A5 P20815 1/20 0.45
CYP2A7 P20853 1/20 0.45
CYP3A7 P24462 1/20 0.45
CYP2F1 P24903 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16890383 0.89 PGR (0.46) LTA4HCYP2C9CYP2C19MEN1KMT2A
SCHEMBL20101688 0.89 CYP1A2 (0.57) CYP11B1CYP11B2CYP17A1HDAC8CYP1A2
SCHEMBL16561425 0.80 HDAC8 (0.49) CYP11B1CYP11B2CYP17A1HDAC8CYP1A2
SCHEMBL12989388 0.80 CYP11B1 (0.52) CYP11B1CYP11B2CYP17A1HDAC8CYP1A2
SCHEMBL28550067 0.78 CYP1A2 (0.56) CYP1A2CYP2A6CYP3A4CYP2D6CYP2C9
SCHEMBL9781864 0.76 CYP1A2 (0.53) CYP11B1CYP11B2CYP17A1HDAC8CYP1A2
SCHEMBL5286981 0.76 BRD4 (0.55) CYP11B1CYP11B2CYP1A2CYP2A6CYP3A4
SCHEMBL6013084 0.75 L3MBTL1 (0.55) LTA4HCYP1A2CYP2A6CYP2C9CYP2C19
SCHEMBL8125066 0.75 HDAC8 (0.54) CYP11B1CYP11B2HDAC8CYP1A2CYP2A6
SCHEMBL3598954 0.75 ALDH1A1 (0.56) CYP1A2CYP3A4CYP2D6CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216285-A1 FLUORESCENT MALEIMIDES AND USES THEREOF Ciba SC Holding AG (CH) 2002-06-26 EP disclosed
WO-2001019939-A1 FLUORESCENT MALEIMIDES AND USES THEREOF CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2001-03-22 WO disclosed