SCHEMBL7704803

SCHEMBL7704803

Nc1cc(-c2ccccc2F)c(N2CCC3(CC2)OCCO3)cc1NC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
PTPN11 Q06124 1/20 0.41
MAPT P10636 3/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
USP2 O75604 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
THRB P10828 1/20 0.40
ALOX15 P16050 1/20 0.40
FPR1 P21462 1/20 0.40
CASP1 P29466 1/20 0.40
PTPN7 P35236 1/20 0.40
BRCA1 P38398 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7138095 0.87 ALDH1A1 (0.37) ALDH1A1PTPN11MAPTKDM4ESMN1; SMN2
SCHEMBL7700624 0.85 HDAC2 (0.46) ALDH1A1NPC1RAB9AMAPK8MAPK10
SCHEMBL7707281 0.85 SMN1; SMN2 (0.45) ALDH1A1MAPTKDM4ESMN1; SMN2L3MBTL1
SCHEMBL7140985 0.73 ALDH1A1 (0.44) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL7143760 0.72 HDAC2 (0.44) ALDH1A1RAB9ALMNA
SCHEMBL14336963 0.68 ALDH1A1 (0.45) ALDH1A1MAPTKDM4ESMN1; SMN2MEN1
SCHEMBL6611884 0.68 HDAC1 (0.40) MAPTKDM4ESMN1; SMN2L3MBTL1NPC1
SCHEMBL6608182 0.68 TSHR (0.48) ALDH1A1MAPTKDM4ESMN1; SMN2L3MBTL1
SCHEMBL7141070 0.67 PTPN11 (0.37) ALDH1A1PTPN11MAPTKDM4ESMN1; SMN2
SCHEMBL23536222 0.66 LGMN (0.58) ALDH1A1PTPN11MAPTKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed