SCHEMBL7704830

SCHEMBL7704830

CC1=C(N)Nc2cc(CN(C(=O)OC(C)(C)C)C3Cc4ccccc4C3)ccc2O1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.35
NR1H4 Q96RI1 1/20 0.33
KDM1A O60341 1/20 0.32
CETP P11597 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
NCOR2 Q9Y618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705016 0.86 RAMP1 (0.35) HSD11B1KDM1A
SCHEMBL7704910 0.82 HDAC1 (0.45) HDAC3HDAC1HDAC2NCOR2
SCHEMBL7710997 0.80 PARP1 (0.36) HSD11B1NR1H4CETPSLC6A2SLC6A4
SCHEMBL7711366 0.79 HDAC1 (0.37) HDAC3HDAC1HDAC2NCOR2
SCHEMBL7708189 0.79 HDAC3 (0.37) HDAC3HDAC1HDAC2NCOR2
SCHEMBL7704988 0.78 HDAC3 (0.36) HDAC3HDAC1HDAC2NCOR2
SCHEMBL7710867 0.78 ALDH1A1 (0.38) HDAC3HDAC1HDAC2NCOR2
SCHEMBL7711307 0.78 ALDH1A1 (0.42)
SCHEMBL7000559 0.78 HDAC1 (0.33) NR1H4SLC6A4HDAC1
SCHEMBL7711360 0.78 TRPM8 (0.36) CETPHDAC3HDAC1HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed