SCHEMBL7710997

SCHEMBL7710997

CC1Oc2ccc(CN(C(=O)OC(C)(C)C)C3Cc4ccccc4C3)cc2NC1=S

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.36
HSD11B1 P28845 1/20 0.35
NR1H4 Q96RI1 1/20 0.33
CETP P11597 1/20 0.31
ALOX15 P16050 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
NCOR2 Q9Y618 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704973 0.86 RAMP1 (0.35) PARP1HSD11B1
SCHEMBL7704884 0.85 P2RX3 (0.40) PARP1ALDH1A1
SCHEMBL7704945 0.83 HDAC3 (0.44) PARP1ALOX15HSD17B10HDAC3HDAC1
SCHEMBL6309617 0.81 HDAC1 (0.43) PARP1ALOX15HSD17B10HDAC3HDAC1
SCHEMBL7710837 0.80 PARP1 (0.40) PARP1ALOX15HSD17B10HDAC3HDAC1
SCHEMBL7704830 0.80 HSD11B1 (0.35) HSD11B1NR1H4CETPSLC6A2SLC6A4
SCHEMBL7704907 0.79 HSD17B10 (0.38) PARP1ALOX15HSD17B10HDAC3HDAC1
SCHEMBL7704942 0.79 ALDH1A1 (0.37) PARP1ALOX15HSD17B10HDAC3HDAC1
SCHEMBL7711006 0.79 PARP1 (0.36) PARP1ALOX15HSD17B10HDAC3HDAC1
SCHEMBL7711323 0.79 ALDH1A1 (0.41) ALOX15HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed