SCHEMBL7705091

SCHEMBL7705091

CC(C)(C)OC(=O)N(C1CCN(Cc2ccccc2)CC1)C(Cc1ccccc1)C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.45
SIGMAR1 Q99720 2/20 0.45
CHRM2 P08172 7/20 0.43
CHRM3 P20309 7/20 0.43
KCNH2 Q12809 1/20 0.43
ACHE P22303 2/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
BCHE P06276 1/20 0.43
OPRD1 P41143 1/20 0.43
OPRK1 P41145 1/20 0.43
CHRM4 P08173 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2494437 0.85 OPRM1 (0.50) OPRM1SIGMAR1CHRM2CHRM3KCNH2
SCHEMBL1205295 0.81 ACHE (0.45) OPRM1SIGMAR1CHRM2CHRM3ACHE
SCHEMBL803672 0.79 SIGMAR1 (0.59) OPRM1SIGMAR1CHRM2CHRM3KCNH2
SCHEMBL34473259 0.79 OPRM1 (0.46) OPRM1SIGMAR1CHRM2CHRM3KCNH2
SCHEMBL65854 0.76 CACNA1B (0.39) ACHEBCHE
SCHEMBL3815654 0.75 SIGMAR1 (0.51) OPRM1SIGMAR1KCNH2ACHEDRD2
SCHEMBL7507555 0.75 SIGMAR1 (0.51) OPRM1SIGMAR1KCNH2ACHEDRD2
SCHEMBL1718867 0.74 CHRM4 (0.53) OPRM1SIGMAR1CHRM2CHRM3KCNH2
SCHEMBL5367694 0.74 OPRM1 (0.54) OPRM1SIGMAR1CHRM2CHRM3KCNH2
SCHEMBL34474746 0.74 CCR5 (0.53) OPRM1SIGMAR1CHRM2CHRM3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344449-B1 HEADACHE AND MORPHINE DEPENDENCE DR. KARL THOMAE GMBH (DE) 2002-02-05 US disclosed