SCHEMBL7704052

SCHEMBL7704052

CN(C)c1ccnc(C2=NCCc3ccccc32)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.45
GRIN3B O60391 1/20 0.45
CHRM1 P11229 1/20 0.45
ADRA1D P25100 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
GRIN1 Q05586 1/20 0.45
GRIN2A Q12879 1/20 0.45
GRIN2B Q13224 1/20 0.45
GRIN2C Q14957 1/20 0.45
GRIN3A Q8TCU5 1/20 0.45
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41
MAOA P21397 2/20 0.39
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
SIRT2 Q8IXJ6 4/20 0.36
PKM P14618 1/20 0.36
RAD52 P43351 1/20 0.36
MAPK10 P53779 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705661 0.79 NOS3 (0.44) NOS3NOS2MAOAKDM4EALDH1A1
SCHEMBL7705872 0.79 MAOA (0.52) NOS3NOS2MAOAALDH1A1PKM
SCHEMBL7701012 0.79 NOS3 (0.49) ADRA1DADRA1AADRA1BNOS3NOS2
SCHEMBL7705613 0.75 NOS3 (0.45) CHRM1ADRA1DADRA1AADRA1BNOS3
SCHEMBL13360717 0.72 CYP1A2 (0.57) GRIN2DGRIN3BCHRM1ADRA1DADRA1A
SCHEMBL196641 0.72 ALDH1A1 (0.53) GRIN2DGRIN3BCHRM1ADRA1DADRA1A
SCHEMBL7697911 0.72 NOS3 (0.45) NOS3NOS2MAOAKDM4EALDH1A1
SCHEMBL7705902 0.70 NOS3 (0.46) CHRM1NOS3NOS2MAOAKDM4E
SCHEMBL30636788 0.70 KDM4E (0.54) GRIN2DGRIN3BCHRM1ADRA1DADRA1A
SCHEMBL30345721 0.70 ASIC3 (0.53) GRIN2DGRIN3BCHRM1ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1098260-C 2,4-diaminopyrimidine derivatives BASLIR PHARMACEUTICALS AG (CH) 2003-01-08 CN disclosed
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
CN-1218465-A 2,4-diaminopyrimidine derivatives HOFFMANN LA ROCHE (CH) 1999-06-02 CN disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed