SCHEMBL7705964

SCHEMBL7705964

[O-][n+]1ccc2nc3ccncc3cc2c1

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 1/20 0.36
CSNK1E P49674 1/20 0.36
CLK1 P49759 1/20 0.36
DYRK1A Q13627 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL255425 0.79 CLK1 (0.48) CSNK1DCSNK1ECLK1DYRK1A
SCHEMBL2989390 0.76 PRKCZ (0.35) CSNK1DCSNK1ECLK1DYRK1A
SCHEMBL2986767 0.76 CYP19A1 (0.33) CSNK1DCSNK1ECLK1DYRK1A
SCHEMBL20272949 0.73 CLK1 (0.53) CSNK1DCSNK1ECLK1DYRK1A
SCHEMBL30520081 0.71 CLK1 (0.47) CSNK1DCSNK1ECLK1DYRK1A
SCHEMBL5894666 0.71 KDM4E (0.33) CSNK1DCSNK1ECLK1DYRK1A
Isoquinoline SCHEMBL5264460 0.70 ACHE (0.37)
SCHEMBL2385144 0.70 ALDH1A1 (0.65) CSNK1DCSNK1ECLK1DYRK1A
SCHEMBL31187649 0.69 EGFR (0.48)
SCHEMBL5894084 0.64 KDM4E (0.31) CSNK1DCSNK1ECLK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169932-B2 HIV protease inhibitors, compositions containing the same, their pharmaceutical uses, material for their synthesis PFIZER INC. (US) 2007-01-30 US disclosed
US-6610730-B2 Viricides; protease inbhibitor AGOURON PHARMACEUTICALS, INC. 2003-08-26 US disclosed