SCHEMBL7706352

SCHEMBL7706352

NC(=O)c1cccc2nc(C3CCN(CCc4ccc(I)cc4)CC3)[nH]c12

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.55
PARP2 Q9UGN5 3/20 0.52
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR7 P34969 1/20 0.42
HTR6 P50406 1/20 0.42
LTA4H P09960 1/20 0.40
HTR2B P41595 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705626 0.91 PARP1 (0.56) PARP1PARP2LTA4H
SCHEMBL7702685 0.90 PARP1 (0.55) PARP1PARP2LTA4H
SCHEMBL7706397 0.90 PARP1 (0.55) PARP1PARP2HTR2CHTR7HTR2B
SCHEMBL7700398 0.90 PARP1 (0.55) PARP1PARP2HTR2B
SCHEMBL7705624 0.90 PARP1 (0.55) PARP1PARP2HTR2AHTR2CHTR7
SCHEMBL7702702 0.88 PARP1 (0.55) PARP1PARP2
SCHEMBL7706364 0.88 PARP1 (0.53) PARP1PARP2HTR2CHTR7LTA4H
SCHEMBL5620912 0.88 PARP1 (0.53) PARP1PARP2
SCHEMBL7705471 0.87 PARP1 (0.62) PARP1PARP2LTA4H
SCHEMBL7706390 0.87 PARP1 (0.52) PARP1PARP2HTR2AHTR7HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed