SCHEMBL7706364

SCHEMBL7706364

COc1ccc(CCN2CCC(c3nc4cccc(C(N)=O)c4[nH]3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.53
PARP2 Q9UGN5 1/20 0.52
KCNH2 Q12809 1/20 0.49
TACR2 P21452 1/20 0.47
TACR1 P25103 1/20 0.47
HRH1 P35367 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
POLB P06746 1/20 0.46
CHEK1 O14757 1/20 0.46
AURKA O14965 1/20 0.46
PRKD3 O94806 1/20 0.46
PAK4 O96013 1/20 0.46
NTRK1 P04629 1/20 0.46
FYN P06241 1/20 0.46
RET P07949 1/20 0.46
MET P08581 1/20 0.46
PDGFRB P09619 1/20 0.46
PIM1 P11309 1/20 0.46
PDGFRA P16234 1/20 0.46
PRKACA P17612 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708486 0.96 PARP1 (0.58) PARP1PARP2KCNH2TACR2TACR1
SCHEMBL7706397 0.90 PARP1 (0.55) PARP1PARP2HRH1HTR2BHTR1A
SCHEMBL5621735 0.89 PARP1 (0.51) PARP1PARP2KCNH2HRH1CHEK1
SCHEMBL7705626 0.89 PARP1 (0.56) PARP1PARP2KCNH2LTA4H
SCHEMBL7702685 0.88 PARP1 (0.55) PARP1PARP2LTA4H
SCHEMBL7700398 0.88 PARP1 (0.55) PARP1PARP2HTR2B
SCHEMBL7706352 0.88 PARP1 (0.55) PARP1PARP2HTR2BHTR2CHTR7
SCHEMBL7705624 0.88 PARP1 (0.55) PARP1PARP2KCNH2TACR2TACR1
SCHEMBL5620233 0.86 PARP1 (0.72) PARP1PARP2CHEK1AURKAPRKD3
SCHEMBL7706345 0.86 PARP1 (0.61) PARP1PARP2HRH1HTR2BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed