SCHEMBL7708206

SCHEMBL7708206

CC1Oc2ccc(CN(C(=O)OC(C)(C)C)C3CCCc4ccccc43)cc2NC1=O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.42
P2RX3 P56373 2/20 0.41
P2RX2 Q9UBL9 2/20 0.41
SMYD3 Q9H7B4 2/20 0.37
TAS2R14 Q9NYV8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
XBP1 P17861 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704884 0.91 P2RX3 (0.40) PARP1P2RX3P2RX2TAS2R14ALDH1A1
SCHEMBL7704973 0.86 RAMP1 (0.35) PARP1P2RX3P2RX2SMYD3TAS2R14
SCHEMBL6608132 0.81 CREBBP (0.39) PARP1P2RX3P2RX2SMYD3
SCHEMBL7705016 0.78 RAMP1 (0.35) P2RX3P2RX2SMN1; SMN2
SCHEMBL7713376 0.77 PARP1 (0.56) PARP1SMYD3ALDH1A1HTTSMN1; SMN2
SCHEMBL6305893 0.76 PARP1 (0.54) PARP1SMYD3ALDH1A1HTTSMN1; SMN2
SCHEMBL7710997 0.75 PARP1 (0.36) PARP1ALDH1A1
SCHEMBL6998344 0.75 PARP1 (0.45) PARP1SMYD3PDE3BPDE3A
SCHEMBL7711130 0.74 PARP1 (0.53) PARP1SMYD3ALDH1A1HTTHTR1A
SCHEMBL6281965 0.74 TMEM97 (0.32) PARP1SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed