SCHEMBL7704973

SCHEMBL7704973

CC1Oc2ccc(CN(C(=O)OC(C)(C)C)C3CCc4ccccc43)cc2NC1=S

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAMP1 O60894 6/20 0.35
CALCRL Q16602 6/20 0.35
P2RX3 P56373 2/20 0.34
P2RX2 Q9UBL9 2/20 0.34
PARP1 P09874 3/20 0.33
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
TAS1R2 Q8TE23 1/20 0.31
HSD11B1 P28845 1/20 0.31
TAS2R14 Q9NYV8 1/20 0.31
SMYD3 Q9H7B4 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704884 0.95 P2RX3 (0.40) RAMP1CALCRLP2RX3P2RX2PARP1
SCHEMBL7710997 0.86 PARP1 (0.36) PARP1HSD11B1
SCHEMBL7708206 0.86 PARP1 (0.42) P2RX3P2RX2PARP1TAS2R14SMYD3
SCHEMBL7705016 0.82 RAMP1 (0.35) RAMP1CALCRLP2RX3P2RX2HSD11B1
SCHEMBL7704945 0.79 HDAC3 (0.44) PARP1SMN1; SMN2
SCHEMBL6309617 0.77 HDAC1 (0.43) PARP1SMN1; SMN2
SCHEMBL6611314 0.76 BRD4 (0.37) P2RX3P2RX2PARP1
SCHEMBL7710837 0.76 PARP1 (0.40) PARP1
SCHEMBL7704907 0.75 HSD17B10 (0.38) PARP1SMN1; SMN2
SCHEMBL7704942 0.75 ALDH1A1 (0.37) PARP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed