SCHEMBL7708407

SCHEMBL7708407

CCOc1cccc(-c2cc(N)n3nc(-c4ccc(Br)o4)nc3c2)c1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.53
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 3/20 0.42
ALDH1A1 P00352 2/20 0.42
RECQL P46063 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
S1PR1 P21453 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703022 0.89 NPC1 (0.56) ADORA2ANPC1RAB9ATP53MAPT
SCHEMBL7705941 0.85 ADORA2A (0.51) ADORA2AALDH1A1
SCHEMBL7703126 0.83 ADORA2A (0.53) ADORA2ANPC1RAB9AMAPTALDH1A1
SCHEMBL7709143 0.83 RXRA (0.44) ADORA2ANPC1RAB9ATP53MAPT
SCHEMBL7703024 0.79 ADORA2A (0.49) ADORA2AALDH1A1TDP1
SCHEMBL7705869 0.78 ADORA2A (0.56) ADORA2ANPC1RAB9ATP53MAPT
SCHEMBL7487041 0.78 ADORA2A (0.51) ADORA2ANPC1RAB9ATP53MAPT
SCHEMBL7708821 0.76 ADORA2A (0.54) ADORA2AMAPTTDP1
SCHEMBL7711821 0.76 ADORA2A (0.54) ADORA2AMAPTALDH1A1MEN1KMT2A
SCHEMBL7708427 0.75 ADORA2A (0.53) ADORA2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed