SCHEMBL7708909

SCHEMBL7708909

Nc1cc(NCc2ccccc2)cc2nc(-c3ccccn3)nn12

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.52
KLKB1 P03952 11/20 0.50
KLK1 P06870 2/20 0.50
F2 P00734 5/20 0.47
F10 P00742 4/20 0.47
NPC1 O15118 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PDE5A O76074 1/20 0.46
CSNK1D P48730 2/20 0.45
HIF1A Q16665 1/20 0.45
KDM4E B2RXH2 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
F12 P00748 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705606 0.85 CSNK1D (0.55) F2NPC1MEN1KMT2ACSNK1D
SCHEMBL7709116 0.84 ADORA2A (0.48) ADORA2AKLKB1F2F10NPC1
SCHEMBL7703131 0.82 ADORA2A (0.46) ADORA2AKLKB1F2F10NPC1
SCHEMBL6867628 0.81 ADORA2A (0.60) ADORA2AKLKB1KLK1F2F10
SCHEMBL7711803 0.81 F2 (0.47) ADORA2AF2CSNK1DKDM4E
SCHEMBL7703034 0.79 CSNK1D (0.53) ADORA2AMEN1KMT2ACSNK1D
SCHEMBL7428533 0.77 ADORA2A (0.60) ADORA2AF2NPC1MEN1KMT2A
SCHEMBL7708668 0.76 PDE5A (0.49) ADORA2APDE5ACSNK1DHIF1A
SCHEMBL7438035 0.76 ADORA2A (0.59) ADORA2AF2NPC1MEN1KMT2A
SCHEMBL6867942 0.76 ADORA2A (0.71) ADORA2AF2KDM4EF12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed