SCHEMBL7708668

SCHEMBL7708668

Nc1cc(NCc2cccc(Cl)c2)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.49
CSNK1D P48730 4/20 0.48
APP P05067 2/20 0.46
ADORA3 P0DMS8 2/20 0.44
ADORA1 P30542 1/20 0.44
HIF1A Q16665 1/20 0.44
FYN P06241 2/20 0.43
KCNN3 Q9UGI6 1/20 0.42
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
NOS2 P35228 1/20 0.42
PDE2A O00408 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ADORA2A P29274 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705606 0.90 CSNK1D (0.55) CSNK1DMAPTTP53
SCHEMBL7703034 0.83 CSNK1D (0.53) CSNK1DAPPADORA1MAPTADORA2A
SCHEMBL7708909 0.76 ADORA2A (0.52) PDE5ACSNK1DHIF1AADORA2A
SCHEMBL7711803 0.76 F2 (0.47) CSNK1DADORA3ADORA1MAPTHDAC1
SCHEMBL7705858 0.75 MAPT (0.46) PDE5ACSNK1DKCNN3MAPTTP53
SCHEMBL7708996 0.72 ADORA3 (0.51) CSNK1DADORA3ADORA1HIF1AMAPT
SCHEMBL7423524 0.70 ALDH1A1 (0.53) CSNK1DADORA3ADORA1MAPTTP53
SCHEMBL6873157 0.70 HPGDS (0.51) CSNK1DPDE2AADORA2ALMNA
SCHEMBL1196472 0.69 MAOB (0.56) PDE5AAPPHIF1AMAPTHDAC6
SCHEMBL7709009 0.69 NPC1 (0.44) ADORA3ADORA1KCNN3MAPTADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed