SCHEMBL7710901

SCHEMBL7710901

Cc1c(S(=O)(=O)Cc2ccccc2)c2ccccn2c1CC(=O)N(C)Cc1ccc(F)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 7/20 1.00
HCRTR1 O43613 6/20 1.00
KMT2A Q03164 1/20 0.44
MAPT P10636 2/20 0.44
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TSPO P30536 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
PTGDR Q13258 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709453 0.98 HCRTR2 (1.00) HCRTR2HCRTR1KMT2AMAPTNPC1
SCHEMBL7707423 0.94 HCRTR2 (1.00) HCRTR2HCRTR1KMT2AMAPTNPC1
SCHEMBL7701854 0.93 HCRTR2 (0.86) HCRTR2HCRTR1KMT2AMAPTNPC1
SCHEMBL7709056 0.90 HCRTR2 (0.82) HCRTR2HCRTR1KMT2AMAPTALDH1A1
SCHEMBL2594270 0.86 HCRTR2 (0.75) HCRTR2HCRTR1KMT2AMAPTNPC1
SCHEMBL7707649 0.85 HCRTR2 (0.82) HCRTR2HCRTR1MAPTALDH1A1LMNA
SCHEMBL7707551 0.83 HCRTR2 (0.71) HCRTR2HCRTR1KMT2AMAPTALDH1A1
SCHEMBL2588741 0.81 HCRTR2 (0.71) HCRTR2HCRTR1KMT2AMAPTNPC1
SCHEMBL2585096 0.80 HCRTR2 (0.74) HCRTR2HCRTR1KMT2AMAPTL3MBTL1
SCHEMBL7709292 0.79 HCRTR2 (1.00) HCRTR2HCRTR1KMT2AMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138266-A1 INDOLIZINE AND IMIDAZOPYRIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed