SCHEMBL7713085

SCHEMBL7713085

COC(=O)c1ccc(C#CC(O)c2ccc3c(c2)C(C)(C)CCS3)cc1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 10/20 0.45
RARB P10826 10/20 0.45
RARG P13631 10/20 0.45
CYP3A4 P08684 3/20 0.45
KMT2A Q03164 1/20 0.45
CYP26A1 O43174 2/20 0.44
RXRA P19793 2/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK4 Q16654 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
PTPN11 Q06124 1/20 0.31
MYC P01106 1/20 0.31
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7715173 0.93 RARA (0.40) RARARARBRARGCYP3A4KMT2A
SCHEMBL7713266 0.90 RARA (0.51) RARARARBRARGCYP3A4KMT2A
SCHEMBL8440028 0.87 RARA (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL7715088 0.87 RARA (0.56) RARARARBRARGCYP3A4KMT2A
SCHEMBL7714935 0.86 RARB (0.42) RARARARBRARGCYP3A4CYP26A1
SCHEMBL7940029 0.83 PDK2 (0.36) RARARARBRARGCYP3A4CYP26A1
SCHEMBL7709298 0.82 RARB (0.44) RARARARBRARGCYP3A4KMT2A
SCHEMBL7714846 0.81 RARA (0.52) RARARARBRARGCYP3A4KMT2A
SCHEMBL7928435 0.80 PDK2 (0.35) RARARARBRARGCYP3A4CYP26A1
SCHEMBL7709227 0.79 CYP3A4 (0.59) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US claimed
EP-0661258-B1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CIRD GALDERMA (FR) 1998-04-08 EP claimed
US-6368608-B1 SKIN DISORDERS CENTRE INTERNATIONAL DE RECHERCHE DERMATOLOGIQUES GALDERMA (C.I.R.D.) (FR) 2002-04-09 US disclosed
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US disclosed