SCHEMBL7709227

SCHEMBL7709227

CC1(C)CCSc2ccc(C(O)C#Cc3ccc(C(=O)O)cc3)cc21

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.59
CYP26A1 O43174 3/20 0.59
RARB P10826 16/20 0.53
RARG P13631 16/20 0.53
RARA P10276 15/20 0.53
RXRA P19793 4/20 0.53
CRABP2 P29373 1/20 0.48
KMT2A Q03164 1/20 0.48
RXRB P28702 1/20 0.45
CYP26B1 Q9NR63 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7713109 0.95 CYP3A4 (0.66) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL7709286 0.92 CYP26A1 (0.52) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL7715088 0.89 RARA (0.56) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL7713266 0.86 RARA (0.51) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL6378967 0.84 RARB (0.68) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9817648 0.84 CYP3A4 (0.76) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8458475 0.83 RXRA (0.68) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8681728 0.81 RARB (0.48) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL7715303 0.81 RARA (0.48) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8101908 0.80 RARB (0.72) CYP3A4CYP26A1RARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US claimed
EP-0661258-B1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CIRD GALDERMA (FR) 1998-04-08 EP claimed
US-6368608-B1 SKIN DISORDERS CENTRE INTERNATIONAL DE RECHERCHE DERMATOLOGIQUES GALDERMA (C.I.R.D.) (FR) 2002-04-09 US disclosed
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US disclosed
EP-0661258-B1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CIRD GALDERMA (FR) 1998-04-08 EP disclosed
EP-0661258-A1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA, ( CIRD GALDERMA) (FR) 1995-07-05 EP disclosed