SCHEMBL7713435

SCHEMBL7713435

CC1=C(N)Nc2cc(CN(Cc3ccc(S(C)(=O)=O)cc3)C(=O)OC(C)(C)C)ccc2O1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.34
HDAC3 O15379 2/20 0.34
HDAC2 Q92769 2/20 0.34
NCOR2 Q9Y618 2/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.32
GPR119 Q8TDV5 4/20 0.31
MAPK8 P45983 2/20 0.30
STAT5B P51692 1/20 0.30
ADRB3 P13945 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7710748 0.93 CA2 (0.35) HDAC1HDAC3HDAC2NCOR2KMT2A
SCHEMBL7708189 0.89 HDAC3 (0.37) HDAC1HDAC3HDAC2NCOR2KMT2A
SCHEMBL7711366 0.89 HDAC1 (0.37) HDAC1HDAC3HDAC2NCOR2ADRB3
SCHEMBL7704910 0.89 HDAC1 (0.45) HDAC1HDAC3HDAC2NCOR2KMT2A
SCHEMBL7708353 0.88 GRM2 (0.37) HDAC1HDAC3HDAC2NCOR2KMT2A
SCHEMBL7704965 0.88 HDAC3 (0.36) HDAC1HDAC3HDAC2NCOR2KMT2A
SCHEMBL7711328 0.87 HDAC3 (0.35) HDAC1HDAC3HDAC2NCOR2KMT2A
SCHEMBL7704946 0.87 ALDH1A1 (0.38) HDAC1HDAC3HDAC2NCOR2
SCHEMBL7708350 0.86 NR1D1 (0.40) HDAC1HDAC3HDAC2NCOR2
SCHEMBL7711458 0.85 HDAC3 (0.33) HDAC1HDAC3HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed