SCHEMBL7713640

SCHEMBL7713640

O=C(O)Cn1nc(S(=O)(=O)Cc2ccccc2)c2ccc(F)cc21

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 3/20 0.54
HCRTR1 O43613 2/20 0.54
PTGDR2 Q9Y5Y4 8/20 0.42
PDE5A O76074 1/20 0.40
HSD17B10 Q99714 1/20 0.40
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.38
CPT1A P50416 1/20 0.38
CPT1B Q92523 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702319 0.94 HCRTR2 (0.47) HCRTR2HCRTR1PTGDR2POLBMAPT
SCHEMBL7707104 0.93 HCRTR1 (0.47) HCRTR2HCRTR1PTGDR2PDE5AHSD17B10
SCHEMBL2595050 0.88 HCRTR2 (0.53) HCRTR2HCRTR1PTGDR2PDE5APOLB
SCHEMBL7707974 0.86 HCRTR2 (0.53) HCRTR2HCRTR1POLBTSHR
SCHEMBL2594744 0.85 HCRTR1 (0.48) HCRTR2HCRTR1POLBMAPTTSHR
SCHEMBL7702650 0.85 HCRTR2 (0.78) HCRTR2HCRTR1HSD17B10POLBMAPT
SCHEMBL7708626 0.85 HCRTR1 (0.71) HCRTR2HCRTR1PTGDR2HSD17B10POLB
SCHEMBL2588992 0.81 HCRTR2 (0.44) HCRTR2HCRTR1POLBMAPT
SCHEMBL7711206 0.81 HCRTR2 (0.55) HCRTR2HCRTR1POLBMAPT
SCHEMBL2594867 0.81 HCRTR1 (0.45) HCRTR2HCRTR1PTGDR2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138265-A2 INDOLE AND INDAZOLE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed