SCHEMBL7714271

SCHEMBL7714271

O=c1[nH]c(Nc2ccc(F)cc2)ncc1Oc1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 7/20 0.44
POLB P06746 1/20 0.43
MAPT P10636 3/20 0.42
LMNA P02545 1/20 0.42
SCN8A Q9UQD0 2/20 0.38
SCN10A Q9Y5Y9 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PNLIP P16233 1/20 0.37
SCN9A Q15858 3/20 0.37
KCNH2 Q12809 1/20 0.37
SCN5A Q14524 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5207646 0.72 KDM4C (0.41) POLBMAPTLMNACYP1A2CYP2C9
SCHEMBL5202998 0.72 LTA4H (0.57) MAPTCYP1A2CYP2C9CYP2C19SCN9A
SCHEMBL7712456 0.72 MEN1 (0.44) MAPTHTT
Methane SCHEMBL7708438 0.71 KDM4C (0.40) POLBMAPTLMNACYP1A2CYP2C9
SCHEMBL7708436 0.69 LMNA (0.52) POLBLMNANPSR1
SCHEMBL7716750 0.69 KDM4C (0.40) CYP1A2CYP2C9CYP2C19HTTNPSR1
SCHEMBL5175115 0.65 MAOA (0.58) MAPTLMNACYP1A2CYP2C9CYP2C19
SCHEMBL7712513 0.63 HRH4 (0.49) POLBCYP1A2
SCHEMBL7716633 0.63 KMT2A (0.49) CYP1A2CYP2C9CYP2C19HTTNPSR1
SCHEMBL3350998 0.63 SOS1 (0.44) POLBMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US disclosed