SCHEMBL7714536

SCHEMBL7714536

CC(C)c1ccc(Oc2cnc(N)[nH]c2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 7/20 0.41
MCHR1 Q99705 6/20 0.41
LTA4H P09960 1/20 0.40
ICAM1 P05362 1/20 0.39
SELE P16581 1/20 0.39
KDM4C Q9H3R0 5/20 0.39
PNP P00491 1/20 0.38
DHFR P00374 1/20 0.36
AURKA O14965 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202998 0.84 LTA4H (0.57) LTA4HKDM4C
SCHEMBL7712501 0.84 XDH (0.45) LTA4H
SCHEMBL5202653 0.84 TEAD4 (0.42) NPBWR1MCHR1LTA4HICAM1SELE
SCHEMBL5207820 0.82 MAPT (0.43) LTA4HICAM1SELEDHFRAURKA
SCHEMBL7712456 0.81 MEN1 (0.44) LTA4HICAM1SELEAURKA
SCHEMBL5206240 0.80 NOS1 (0.45) LTA4HKDM4C
SCHEMBL5204052 0.80 SMN1; SMN2 (0.42) NPBWR1MCHR1LTA4HICAM1SELE
SCHEMBL5206874 0.77 L3MBTL1 (0.41) LTA4HICAM1SELEKDM4C
SCHEMBL7712398 0.77 TYMS (0.43) LTA4HKDM4C
SCHEMBL5204487 0.74 SOS1 (0.40) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US disclosed