SCHEMBL7715206

SCHEMBL7715206

NC(c1ccccc1)(c1cccc(OC(=O)C(F)(F)F)c1)[C@@H]1CCNC1=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.35
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
PRSS1 P07477 1/20 0.32
ACR P10323 1/20 0.32
GAA P10253 2/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
EPHX2 P34913 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10732623 0.69 PRSS1 (0.52) PRSS1ACRGAAPPARGPPARA
SCHEMBL11370912 0.66 ATM (0.41) PRSS1ACRGAAPPARGPPARA
SCHEMBL1255890 0.65 ELANE (0.47) KDM4EALDH1A1
SCHEMBL4658587 0.65 AKR1C3 (0.51) SMN1; SMN2KMT2AMEN1KDM4EALDH1A1
SCHEMBL10946374 0.64 ELANE (0.46) KDM4EALDH1A1
SCHEMBL7715202 0.63 MGLL (0.38) ALDH1A1
SCHEMBL20528635 0.62 SMN1; SMN2 (0.44) SMN1; SMN2KMT2AMEN1GAALMNA
SCHEMBL10180800 0.62 ESR1 (0.49) KMT2AMEN1PPARGPPARAALDH1A1
SCHEMBL11436506 0.62 CYP3A4 (0.59) KMT2AMEN1ALDH1A1LMNA
SCHEMBL27284217 0.61 PARP1 (0.57) KMT2AMEN1PRSS1ACREPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed