SCHEMBL7715202

SCHEMBL7715202

N[C@H]1CCN(C(c2ccccc2)c2cccc(OC(=O)C(F)(F)F)c2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 7/20 0.38
SLC6A9 P48067 1/20 0.36
USP2 O75604 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
HIF1A Q16665 1/20 0.34
DPP4 P27487 4/20 0.34
DPP7 Q9UHL4 2/20 0.34
OPRM1 P35372 2/20 0.34
OPRD1 P41143 2/20 0.34
OPRK1 P41145 2/20 0.34
OPRL1 P41146 2/20 0.34
NOTUM Q6P988 1/20 0.34
CACNA2D1 P54289 1/20 0.34
CACNA1B Q00975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7713231 0.91 DPP4 (0.41) MGLLDPP4DPP7OPRM1OPRD1
Trifluoroacetic Acid SCHEMBL7718434 0.82 DPP4 (0.40) SLC6A9DPP4DPP7OPRM1OPRD1
SCHEMBL4463788 0.78 DPP4 (0.46) CYP3A4ALDH1A1CYP2D6TSHRDPP4
Trifluoroacetic Acid SCHEMBL7713229 0.74 DPP4 (0.48) DPP4DPP7OPRM1OPRD1OPRK1
SCHEMBL10331845 0.68 ACE (0.52) CYP3A4ALDH1A1TSHRDPP4
SCHEMBL1255890 0.65 ELANE (0.47) ALDH1A1
SCHEMBL4658587 0.64 AKR1C3 (0.51) ALDH1A1
SCHEMBL10946374 0.63 ELANE (0.46) ALDH1A1
SCHEMBL7715206 0.63 SMN1; SMN2 (0.35) ALDH1A1
SCHEMBL1527357 0.62 ALDH1A1 (0.51) CYP3A4ALDH1A1CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed