SCHEMBL7719892

SCHEMBL7719892

O=C(Cc1ccccc1-c1ccccn1)N[C@H]1CCN(CCc2ccc(F)cc2)C1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 11/20 0.52
CCR3 P51677 4/20 0.46
NPC1 O15118 1/20 0.44
PRCP P42785 1/20 0.43
ALDH1A1 P00352 1/20 0.42
CCR5 P51681 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7719896 1.00 SIGMAR1 (0.52) SIGMAR1CCR3NPC1PRCPALDH1A1
SCHEMBL7729788 0.92 SIGMAR1 (0.57) SIGMAR1
SCHEMBL7729790 0.92 SIGMAR1 (0.57) SIGMAR1
SCHEMBL7729835 0.79 SIGMAR1 (0.56) SIGMAR1CCR3NPC1CCR5
SCHEMBL7729841 0.79 SIGMAR1 (0.56) SIGMAR1CCR3NPC1CCR5
SCHEMBL7729514 0.77 DRD2 (0.45) SIGMAR1CCR3
SCHEMBL7729521 0.77 DRD2 (0.45) SIGMAR1CCR3
SCHEMBL6618321 0.74 NOS1 (0.55) SIGMAR1CCR3CCR5
SCHEMBL31486979 0.71 SIGMAR1 (0.71) SIGMAR1CCR3
SCHEMBL7719812 0.71 NR4A2 (0.48) SIGMAR1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6468998-B1 ANTAGONIZE SEROTONIN 2 RECEPTORS, SUPPRESS PLATELET AGGREGATION, IMPROVE PERIPHERAL CIRCULATION AND PROMOTE LACHRYMATION MITSUBISHI PHARMA CORPORATION (JP) 2002-10-22 US disclosed
EP-1125922-A1 PYRROLIDINE COMPOUNDS AND MEDICINAL UTILIZATION THEREOF Welfide Corporation (JP) 2001-08-22 EP disclosed