Triaziquone

Triaziquone

SCHEMBL7720256

CC(N)N.O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 1/20 0.44
MAPT P10636 3/20 0.42
HTT P42858 3/20 0.42
TP53 P04637 1/20 0.42
STAT3 P40763 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TDP2 O95551 3/20 0.38
NSD2 O96028 3/20 0.38
APAF1 O14727 2/20 0.38
HKDC1 Q2TB90 2/20 0.38
KMT2A Q03164 2/20 0.36
ATG4B Q9Y4P1 2/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
GALK1 P51570 1/20 0.36
BLM P54132 1/20 0.36
ATM Q13315 1/20 0.36
NOD2 Q9HC29 1/20 0.36
LMNA P02545 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL322828 0.93 DNMT1 (0.42) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL149876 0.90 MAPT (0.46) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL10567262 0.90 DNMT1 (0.40) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL3100107 0.89 DNMT1 (0.44) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL8303 0.88 DNMT1 (0.48) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL4612122 0.88 DNMT1 (0.41) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL8333670 0.87 DNMT1 (0.38) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL10906735 0.87 HTT (0.43) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL11039269 0.87 MAPT (0.43) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL7783197 0.86 MAPT (0.46) DNMT1MAPTHTTTP53STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4087676-A1 SUBMICRON PUU-CAPSULES AND MANUFACTURING THEREOF EMPA Eidgenössische Materialprüfungs- und Forschungsanstalt (CH) 2022-11-16 EP disclosed
WO-2021144454-A1 SUBMICRON PUU-CAPSULES AND MANUFACTURING THEREOF EMPA EIDGENÖSSISCHE MATERIALPRÜFUNGS- UND FORSCHUNGSANSTALT (CH) 2021-07-22 WO disclosed
EP-3484973-A1 ADHESIVE DUAL-COMPONENT COMPOSITION BASED ON POLYURETHANE Bostik SA (FR) 2019-05-22 EP disclosed
EP-1236473-A2 Self-assembling polynucleotide delivery system THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2002-09-04 EP disclosed
US-6037444-A COMPOUND OR POLYMER HAVING THIOL, HYDROXY, AMINO OR CARBOXYLIC GROUP IS REACTED WITH A COMPOUND COMPRISING AT LEAST TWO FUNCTIONAL GROUPS SELECTED FROM HYDROXYL, THIOL, AMINO AND CARBOXYLIC ACID GROUPS WHICH FUNCTIONAL GROUPS COURTAULDS COATINGS (HOLDINGS) LIMITED (GB) 2000-03-14 US disclosed
EP-0888279-A1 SELECTIVE CHEMICAL REACTIONS AND POLYMERS OF CONTROLLED ARCHITECTURE PRODUCED THEREBY COURTAULDS COATINGS (HOLDINGS) LIMITED (GB) 1999-01-07 EP disclosed
EP-0636028-A4 SELF-ASSEMBLING POLYNUCLEOTIDE DELIVERY SYSTEM. UNIV CALIFORNIA (US) 1998-12-09 EP disclosed
WO-1997023443-A1 SELECTIVE CHEMICAL REACTIONS AND POLYMERS OF CONTROLLED ARCHITECTURE PRODUCED THEREBY COURTAULDS COATINGS (HOLDINGS) LIMITED (GB) 1997-07-03 WO disclosed
US-5565184-A Functionalized tripodal ligands for x-ray & radioactive imaging applications MALLINCKRODT MEDICAL, INC. (US) 1996-10-15 US disclosed
EP-0664819-A1 CHELATING POLYMERS. STERLING WINTHROP INC (US) 1995-08-02 EP disclosed
EP-0664714-A1 MR IMAGING COMPOSITIONS, BASED ON POLY(ALKYLENEOXIDE) NYCOMED IMAGING AS (NO) 1995-08-02 EP disclosed
EP-0664713-A1 THERAPEUTIC AND DIAGNOSTIC IMAGING COMPOSITIONS AND METHODS NYCOMED IMAGING AS (NO) 1995-08-02 EP disclosed
EP-0636028-A1 SELF-ASSEMBLING POLYNUCLEOTIDE DELIVERY SYSTEM THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-02-01 EP disclosed
WO-1994008624-A2 THERAPEUTIC AND DIAGNOSTIC IMAGING COMPOSITIONS AND METHODS STERLING WINTHROP INC. (US) 1994-04-28 WO disclosed
WO-1994009056-A1 CHELATING POLYMERS STERLING WINTHROP INC. (US) 1994-04-28 WO disclosed
WO-1994008629-A1 MR IMAGING COMPOSITIONS, BASED ON POLY(ALKYLENEOXIDE) STERLING WINTHROP INC. (US) 1994-04-28 WO disclosed
WO-1993019768-A1 SELF-ASSEMBLING POLYNUCLEOTIDE DELIVERY SYSTEM THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1993-10-14 WO disclosed