SCHEMBL7720962

SCHEMBL7720962

COc1cc(OC)c2c(CN)ncc(NC(=O)N(C)Cc3ccccc3)c2c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.49
ABCC1 P33527 1/20 0.43
HTT P42858 3/20 0.41
TSHR P16473 2/20 0.41
ALOX15 P16050 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
ROCK2 O75116 3/20 0.39
ROCK1 Q13464 2/20 0.39
CYP2C9 P11712 1/20 0.39
CDC42BPA Q5VT25 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362219 0.91 GAA (0.49) DPP4HTTTSHRSMN1; SMN2GAA
SCHEMBL3362425 0.89 DPP4 (0.50) DPP4HTTTSHRALOX15SMN1; SMN2
SCHEMBL3361478 0.89 DPP4 (0.45) DPP4ABCC1HTTSMN1; SMN2GAA
SCHEMBL3363078 0.86 DPP4 (0.58) DPP4
SCHEMBL3362038 0.85 DPP4 (0.57) DPP4ABCC1HTTTSHRALOX15
SCHEMBL7716634 0.85 ABCC1 (0.38) DPP4ABCC1HTTTSHRALOX15
SCHEMBL3363889 0.84 DPP4 (0.59) DPP4HTTGAAMAPK1ROCK2
SCHEMBL3361996 0.81 DPP4 (0.49) DPP4HTTTSHRSMN1; SMN2GAA
SCHEMBL3361319 0.77 GAA (0.44) HTTSMN1; SMN2GAAMAPK1MEN1
SCHEMBL3363084 0.77 DPP4 (0.53) DPP4HTTGAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed