SCHEMBL7724616

SCHEMBL7724616

O=C(O)C1CSC(c2ccccc2OCc2ccccc2)=N1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.50
RXRB P28702 1/20 0.50
RXRG P48443 1/20 0.50
HTR2B P41595 1/20 0.46
MCL1 Q07820 1/20 0.45
PTGER1 P34995 10/20 0.44
PTGER4 P35408 7/20 0.44
PTGER3 P43115 7/20 0.44
PTGER2 P43116 7/20 0.44
DRD2 P14416 1/20 0.43
DRD1 P21728 1/20 0.43
TBXA2R P21731 1/20 0.43
DRD4 P21917 1/20 0.43
DRD5 P21918 1/20 0.43
DRD3 P35462 1/20 0.43
PTGFR P43088 1/20 0.43
PTGIR P43119 1/20 0.43
IDO1 P14902 1/20 0.43
BRD4 O60885 2/20 0.41
ERN1 O75460 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15602818 0.91 RXRA (0.43) RXRARXRBRXRGHTR2BMCL1
SCHEMBL4556877 0.76 RXRA (0.51) RXRARXRBRXRGMCL1PTGER1
SCHEMBL30608416 0.76 HTR2B (0.76) HTR2B
SCHEMBL1534272 0.76 HTR2B (0.76) HTR2B
SCHEMBL1686982 0.76 HTR2B (0.76) HTR2B
SCHEMBL7723380 0.75 RXRA (0.50) RXRARXRBRXRGMCL1PTGER1
SCHEMBL7724707 0.75 RXRA (0.50) RXRARXRBRXRGMCL1PTGER1
SCHEMBL5999284 0.74 HTR2B (0.54) HTR2B
SCHEMBL1268161 0.73 HTR2B (0.47) HTR2BERN1
SCHEMBL15602761 0.73 ALDH1A1 (0.47) HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403623-B1 ADMINISTERING 2-(2-SUBSTITUTED-PHENYL)-2-OXAZOLINES AND RELATED 5-MEMBERED HETEROCYCLES UNUVERSITY OF NOTRE DAME DU LAC 2002-06-11 US claimed
US-6403623-B1 ADMINISTERING 2-(2-SUBSTITUTED-PHENYL)-2-OXAZOLINES AND RELATED 5-MEMBERED HETEROCYCLES UNUVERSITY OF NOTRE DAME DU LAC 2002-06-11 US disclosed
US-6310058-B1 N-HYDROXYAZEPIN-2-ONES SUBSTITUTED AT 3 POSITION WITH A GROUP CONTAINING A 2-PHENYLOXAZOLE OR 2-PHENYLOXAZOLINE GROUP FOR TREATING TUBERCULOSIS UNIVERSITY OF NOTRE DAME DU LAC 2001-10-30 US disclosed