SCHEMBL7729073

SCHEMBL7729073

Cc1cccc(C(=O)Cl)c1.O=C(Cl)c1cccc(C(F)(F)F)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.63
KCNK9 Q9NPC2 1/20 0.63
MEN1 O00255 3/20 0.61
KMT2A Q03164 3/20 0.61
HTT P42858 1/20 0.61
RAB9A P51151 1/20 0.61
CES2 O00748 2/20 0.59
NPSR1 Q6W5P4 1/20 0.51
GAA P10253 1/20 0.50
SRD5A2 P31213 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
ALDH1A1 P00352 3/20 0.49
POLB P06746 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
MAPT P10636 1/20 0.48
ADORA1 P30542 1/20 0.48
HSD17B10 Q99714 1/20 0.48
P2RX1 P51575 1/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethane SCHEMBL27364386 0.90 CES2 (0.67) KCNK3KCNK9MEN1KMT2AHTT
SCHEMBL29425720 0.90 CES2 (0.71) KCNK3MEN1KMT2ACES2NPSR1
SCHEMBL19310 0.90 CES2 (0.71) KCNK3MEN1KMT2ACES2NPSR1
SCHEMBL18371866 0.87 CES2 (0.79) KCNK3KCNK9MEN1KMT2AHTT
SCHEMBL17586586 0.87 KCNK3 (0.67) KCNK3KCNK9MEN1KMT2AHTT
SCHEMBL103438 0.84 PARP1 (0.63) KCNK3KCNK9MEN1KMT2ARAB9A
SCHEMBL29365229 0.84 PARP1 (0.63) KCNK3KCNK9MEN1KMT2ARAB9A
Acetone SCHEMBL27922108 0.79 MEN1 (0.58) KCNK3KCNK9MEN1KMT2AHTT
Benzoyl Chloride SCHEMBL10954201 0.79 SMN1; SMN2 (0.59) KCNK3KCNK9MEN1KMT2ARAB9A
SCHEMBL12055235 0.78 CES2 (0.50) KCNK3KCNK9MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015479-A4 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR LILLY CO ELI (US) 2002-07-24 EP disclosed
EP-1015479-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046631-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed