SCHEMBL7729134

SCHEMBL7729134

COC(=O)[C@H]1C[C@H](N(C(=O)CN)C(=O)OC(C)(C)C)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.38
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.35
AGTR2 P50052 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD11B1 P28845 1/20 0.34
NPC1 O15118 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN3A Q9NY46 1/20 0.34
SCN4A P35499 1/20 0.33
FKBP1A P62942 1/20 0.33
MMP2 P08253 1/20 0.33
ANPEP P15144 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7729049 1.00 PTPN1 (0.38) PTPN1NR1H2NR1H3SMN1; SMN2HSD17B10
SCHEMBL7722056 0.90 HSD17B10 (0.40) SMN1; SMN2HSD17B10AGTR2MEN1KMT2A
SCHEMBL7722230 0.90 HSD17B10 (0.40) SMN1; SMN2HSD17B10AGTR2MEN1KMT2A
SCHEMBL7733526 0.88 PTPN1 (0.39) PTPN1NR1H2NR1H3SMN1; SMN2HSD11B1
SCHEMBL7726393 0.88 PTPN1 (0.39) PTPN1NR1H2NR1H3SMN1; SMN2HSD11B1
SCHEMBL7733813 0.88 PTPN1 (0.39) PTPN1NR1H2NR1H3SMN1; SMN2HSD11B1
SCHEMBL7726101 0.78 HSD17B10 (0.34) PTPN1NR1H2SMN1; SMN2HSD17B10AGTR2
SCHEMBL7728185 0.78 HSD17B10 (0.34) PTPN1NR1H2SMN1; SMN2HSD17B10AGTR2
SCHEMBL7727961 0.78 HSD17B10 (0.34) PTPN1NR1H2SMN1; SMN2HSD17B10AGTR2
SCHEMBL25209424 0.76 MMP2 (0.50) PTPN1NR1H2NR1H3SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed