SCHEMBL7731015

SCHEMBL7731015

CCCCn1c(N)c(NC(=O)/C=C/c2cc(OC)c(OC)c(OC)c2)c(=O)n(CCCC)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.54
HTR2C P28335 2/20 0.54
HTR2A P28223 1/20 0.54
SLC6A4 P31645 1/20 0.54
HTR7 P34969 1/20 0.54
HTR6 P50406 1/20 0.54
TERT O14746 1/20 0.53
ALDH1A1 P00352 7/20 0.52
HTT P42858 2/20 0.46
PSMB11 A5LHX3 1/20 0.46
PSMA7 O14818 1/20 0.46
PSMB1 P20618 1/20 0.46
PSMA1 P25786 1/20 0.46
PSMA2 P25787 1/20 0.46
PSMA3 P25788 1/20 0.46
PSMA4 P25789 1/20 0.46
PSMB8 P28062 1/20 0.46
PSMB9 P28065 1/20 0.46
PSMA5 P28066 1/20 0.46
PSMB4 P28070 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7731020 1.00 HTR1A (0.54) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL7732188 0.94 TERT (0.55) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL7732179 0.94 TERT (0.55) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL7728766 0.83 PSMB11 (0.52) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL7728772 0.83 PSMB11 (0.52) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL7730987 0.83 ADORA2A (0.51) ALDH1A1HTTCA12CA1CA2
SCHEMBL7730989 0.83 ADORA2A (0.51) ALDH1A1HTTCA12CA1CA2
SCHEMBL8372544 0.78 KMT2A (0.51) ALDH1A1CA12CA1CA2CA9
SCHEMBL8372545 0.78 KMT2A (0.51) ALDH1A1CA12CA1CA2CA9
SCHEMBL30632573 0.77 MEN1 (0.52) HTR1AALDH1A1HTTCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628311-B1 Xanthine-Derivatives as Antidepressants KYOWA HAKKO KOGYO KK (JP) 2002-04-24 EP disclosed
EP-0559893-B1 XANTHINE DERIVATIVE KYOWA HAKKO KOGYO KK (JP) 1999-02-03 EP disclosed
US-5543415-A ADMINISTERING A XANTHINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-08-06 US disclosed
EP-0628311-A1 ANTIDEPRESSANT KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-12-14 EP disclosed
EP-0559893-A1 XANTHINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-15 EP disclosed