SCHEMBL7733780

SCHEMBL7733780

Cc1cc(C)c(S(=O)(=O)Cl)c(C)c1.O=S(=O)(Cl)c1ccc(Br)cc1.O=[N+]([O-])c1cccc(S(=O)(=O)Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
ALDH1A1 P00352 3/20 0.46
LMNA P02545 3/20 0.46
MAPK1 P28482 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CA2 P00918 2/20 0.45
CA5A P35218 1/20 0.45
EDNRA P25101 2/20 0.44
EDNRB P24530 1/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TSHR P16473 1/20 0.42
ACHE P22303 1/20 0.42
CA1 P00915 1/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP8 P22894 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8592078 0.87 KMT2A (0.60) KMT2AGAAHTTALDH1A1LMNA
SCHEMBL8093693 0.81 KMT2A (0.53) KMT2AGAAHTTALDH1A1LMNA
SCHEMBL58443 0.79 KMT2A (0.72) KMT2AGAAHTTALDH1A1LMNA
Hydrochloric Acid SCHEMBL7569226 0.77 KMT2A (0.70) KMT2AGAAHTTALDH1A1LMNA
Hydrochloric Acid SCHEMBL7569229 0.77 KMT2A (0.70) KMT2AGAAHTTALDH1A1LMNA
SCHEMBL9143049 0.74 KMT2A (0.66) KMT2AGAAHTTALDH1A1LMNA
SCHEMBL6898125 0.73 ALDH1A1 (0.55) KMT2AHTTALDH1A1LMNAL3MBTL1
SCHEMBL4013923 0.73 RAPGEF4 (0.63) KMT2AGAAHTTALDH1A1L3MBTL1
SCHEMBL11435100 0.71 ALDH1A1 (0.48) KMT2AGAAHTTALDH1A1LMNA
SCHEMBL8664087 0.70 KMT2A (0.80) KMT2AGAAHTTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015479-A4 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR LILLY CO ELI (US) 2002-07-24 EP disclosed
EP-1015479-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
WO-1998046631-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed
WO-1998008839-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED THIOPHENE LIBRARIES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed