SCHEMBL7734067

SCHEMBL7734067

CS(=O)(=O)OCCCc1cn2c3c(cc(F)cc13)CCC2

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.41
MTNR1B P49286 5/20 0.41
HTR2A P28223 3/20 0.39
HTR2C P28335 3/20 0.39
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7734854 0.81 MTNR1A (0.47) MTNR1AMTNR1BHTR2AHTR2C
SCHEMBL6364152 0.76 HTR2A (0.63) MTNR1AMTNR1BHTR2AHTR2C
SCHEMBL5796602 0.65 KDM4E (0.39) MTNR1AMTNR1BHTR2AHTR2C
SCHEMBL5232827 0.63 KDM4E (0.47)
SCHEMBL3899800 0.63 HTR2A (0.43) HTR2AHTR2C
SCHEMBL3702253 0.61 MPO (0.62) HTR2A
SCHEMBL23302470 0.60 PARP1 (0.37)
SCHEMBL3578553 0.59 LMNA (0.45)
SCHEMBL3597833 0.59 KDM4E (0.41)
SCHEMBL5637174 0.59 HTR2A (0.55) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6828325-B2 A benzoxazolopiperazine derivative useful for treating Parkinson's diseases, schizophrenia, anxiety and depression SOLVAY PHARMACEUTICALS B.V. (CH) 2004-12-07 US disclosed