SCHEMBL7736898

SCHEMBL7736898

Cn1cncc1C(CCCN1CCN(S(=O)(=O)c2cccc(O)c2)CC1)(N[S+]([O-])C(C)(C)C)c1ccc(C#N)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.35
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
ERBB2 P04626 1/20 0.33
CCR2 P41597 4/20 0.33
FNTA P49354 5/20 0.32
FNTB P49356 5/20 0.32
PGGT1B P53609 5/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
TRPV4 Q9HBA0 5/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7758000 0.96 PKM (0.33) PKMALDH1A1LMNATSHRKMT2A
SCHEMBL7701717 0.80 FNTB (0.39) FNTAFNTBPGGT1B
SCHEMBL7694904 0.80 FNTB (0.39) FNTAFNTBPGGT1B
SCHEMBL7589567 0.80 FNTB (0.39) FNTAFNTBPGGT1B
Hydrochloric Acid SCHEMBL7757997 0.78 FNTA (0.30) PKMFNTAFNTBPGGT1B
SCHEMBL7736917 0.76 FNTA (0.37) FNTAFNTBPGGT1B
SCHEMBL7582554 0.74 FNTB (0.34) FNTAFNTBPGGT1B
SCHEMBL7700542 0.72 POLB (0.43) ALDH1A1LMNATSHRKMT2AFNTA
SCHEMBL6003297 0.72 POLB (0.43) ALDH1A1LMNATSHRKMT2AFNTA
SCHEMBL7228470 0.70 TRPV4 (0.35) KMT2AFNTAFNTBPGGT1BTRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413964-B1 14-AMINO-14-(1-METHYL-1H-IMIDAZOL-5-YL)-8-OXA-2-THIA-1,18 -DIAZATETRACYCLO(16.2.2.1(3,7).1(9,13))TETRACOSA-3(24),4,6, 9(23),10,12-HEXAENE-10-CARBONITRILE 2,2-DIOXIDE, FOR EXAMPLE; USE IN RADIOTHERAPY, CHEMOTHERAPY AS SENSITIZER MERCK & CO., INC. 2002-07-02 US disclosed
WO-2001051125-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-07-19 WO disclosed