SCHEMBL7738440

SCHEMBL7738440

C=CC[Si](C)(C)c1cc(C[C@H](NC(C)=O)C(=O)OC)c2ccccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.46
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TACR3 P29371 1/20 0.38
HCRTR1 O43613 1/20 0.38
MAPT P10636 3/20 0.36
TP53 P04637 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
NFKB1 P19838 1/20 0.36
APEX1 P27695 1/20 0.36
CYP2C19 P33261 1/20 0.36
THPO P40225 1/20 0.36
BLM P54132 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7738442 1.00 TACR1 (0.46) TACR1MEN1KMT2ATACR3HCRTR1
SCHEMBL7738402 0.77 NOS2 (0.43) TACR1KMT2AALDH1A1POLBCYP2C9
SCHEMBL7738409 0.77 NOS2 (0.43) TACR1KMT2AALDH1A1POLBCYP2C9
SCHEMBL11027965 0.75 TACR1 (0.69) TACR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL11027962 0.75 TACR1 (0.69) TACR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL7738441 0.75 AKR1B1 (0.32) TACR1KDM4EALDH1A1
SCHEMBL7738435 0.73 TAS1R3 (0.33) TACR1ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL7738429 0.73 TAS1R3 (0.33) TACR1ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL7736594 0.71 KDM4E (0.36) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL7736591 0.71 KDM4E (0.36) MEN1KMT2AKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6416861-B1 COMBINATORIAL CHEMISTRY NORTHWESTERN UNIVERSITY 2002-07-09 US disclosed
WO-2000049022-A2 ORGANOSILICON COMPOUNDS AND USES THEREOF NORTHWESTERN UNIVERSITY (US) 2000-08-24 WO disclosed