SCHEMBL7738876

SCHEMBL7738876

Cc1c(NC(=S)NC(=O)c2ccccc2)ccc(-n2cccn2)c1CNC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
MAPT P10636 4/20 0.41
NPSR1 Q6W5P4 3/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
RXFP1 Q9HBX9 1/20 0.41
EPHX1 P07099 3/20 0.40
LMNA P02545 2/20 0.38
MEN1 O00255 5/20 0.38
KMT2A Q03164 5/20 0.38
ALOX12 P18054 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
BLM P54132 1/20 0.37
NAMPT P43490 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7738864 0.87 SYK (0.35) ALDH1A1MAPTNPSR1RAB9ALMNA
SCHEMBL7734198 0.79 TSHR (0.34) ALDH1A1MAPTNPSR1RAB9ALMNA
SCHEMBL7738995 0.79 JAK2 (0.35) LMNAKDM4EMAPK1NAMPT
SCHEMBL29792605 0.70 KLKB1 (0.40) ALDH1A1MAPTMEN1KMT2A
SCHEMBL23118891 0.70 KLKB1 (0.40) ALDH1A1MAPTMEN1KMT2A
SCHEMBL5386906 0.70 ALDH1A1 (0.56) ALDH1A1MAPTNPSR1NPC1RAB9A
SCHEMBL7740422 0.70 SYK (0.40) ALDH1A1MAPTNPSR1RAB9ARXFP1
SCHEMBL7734201 0.69 SYK (0.33) MAPK1
SCHEMBL6757735 0.68 SMN1; SMN2 (0.61) ALDH1A1MAPTNPSR1NPC1RAB9A
SCHEMBL7740426 0.67 PDK1 (0.40) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed