SCHEMBL7738895

SCHEMBL7738895

CCSC(=N)Nc1ccc(-n2cccn2)c(CN)c1C

nearest known ligand 0.32

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
NPC1 O15118 1/20 0.32
MAPK1 P28482 1/20 0.32
ALDH1A1 P00352 5/20 0.31
MEN1 O00255 4/20 0.31
MAPT P10636 4/20 0.31
KMT2A Q03164 4/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
G6PD P11413 1/20 0.31
ADORA2A P29274 1/20 0.31
RAB9A P51151 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7738922 0.99 LMNA (0.32) LMNAHDAC3HDAC1NPC1MAPK1
Hydrochloric Acid SCHEMBL27559416 0.99 LMNA (0.32) LMNAHDAC3HDAC1NPC1MAPK1
Hydrochloric Acid SCHEMBL7742145 0.83 NPC1 (0.33) LMNANPC1MAPK1ALDH1A1MEN1
SCHEMBL7734198 0.80 TSHR (0.34) LMNAHDAC1MAPK1ALDH1A1MEN1
SCHEMBL7739655 0.78 KMT2A (0.36) LMNANPC1MAPK1ALDH1A1MEN1
Hydrochloric Acid SCHEMBL7740465 0.77 KMT2A (0.36) LMNANPC1MAPK1ALDH1A1MEN1
SCHEMBL7738898 0.76 NOS3 (0.40)
SCHEMBL7734196 0.75 HDAC3 (0.32) LMNAHDAC3HDAC1ALDH1A1MEN1
Hydrochloric Acid SCHEMBL7738927 0.75 NOS3 (0.41)
Hydrochloric Acid SCHEMBL7742146 0.67 HCRTR1 (0.32) LMNANPC1MAPK1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN claimed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US claimed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN claimed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP claimed
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed