SCHEMBL7734196

SCHEMBL7734196

CCSC(=N)Nc1ccc(-n2cccn2)c(C(N)C(=O)OC(C)(C)C)c1C

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
TNIK Q9UKE5 1/20 0.32
JAK2 O60674 1/20 0.31
JAK3 P52333 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
MEN1 O00255 3/20 0.31
ALDH1A1 P00352 3/20 0.31
MAPT P10636 3/20 0.31
KMT2A Q03164 3/20 0.31
LMNA P02545 1/20 0.31
RAB9A P51151 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27493987 0.84 ALDH1A1 (0.33) HDAC3HDAC1TNIKJAK2JAK3
SCHEMBL27525664 0.82 RXFP1 (0.35) TNIKRXFP1MEN1ALDH1A1MAPT
SCHEMBL7734198 0.80 TSHR (0.34) HDAC1MEN1ALDH1A1MAPTKMT2A
SCHEMBL7738895 0.75 LMNA (0.32) HDAC3HDAC1MEN1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL7738922 0.74 LMNA (0.32) HDAC3HDAC1MEN1ALDH1A1MAPT
SCHEMBL7740424 0.71 MEN1 (0.36) RXFP1MEN1ALDH1A1MAPTKMT2A
SCHEMBL27564255 0.70 NTRK1 (0.31)
SCHEMBL27495566 0.69 GPR119 (0.35)
SCHEMBL7740420 0.67 SYK (0.37) RXFP1MEN1ALDH1A1MAPTKMT2A
SCHEMBL7738864 0.66 SYK (0.35) HDAC1MEN1ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed