SCHEMBL7739643

SCHEMBL7739643

CCOP(=O)(OCC)c1cc2cc(-c3ccc(F)cc3)c(Cl)cc2[nH]c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.37
CYP1A2 P05177 1/20 0.37
PRKAG1 P54619 5/20 0.37
PRKAA1 Q13131 5/20 0.37
PRKAB1 Q9Y478 5/20 0.37
SSTR2 P30874 1/20 0.36
HSD17B10 Q99714 3/20 0.35
USP2 O75604 1/20 0.35
POLB P06746 1/20 0.35
CASP1 P29466 1/20 0.35
PTPN7 P35236 1/20 0.35
BLM P54132 1/20 0.35
KMT2A Q03164 1/20 0.35
WRN Q14191 1/20 0.35
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7741117 0.90 PRKAG1 (0.37) GSK3BCYP1A2PRKAG1PRKAA1PRKAB1
SCHEMBL7739842 0.89 PRKAG1 (0.42) CYP1A2PRKAG1PRKAA1PRKAB1KMT2A
SCHEMBL7740612 0.89 PRKAG1 (0.40) GSK3BCYP1A2PRKAG1PRKAA1PRKAB1
SCHEMBL7740617 0.89 PTGES (0.36) PRKAG1PRKAA1PRKAB1GRIN2DGRIN3B
SCHEMBL7741113 0.86 IDH1 (0.41) PRKAG1PRKAA1PRKAB1GRIN2DGRIN3B
SCHEMBL7742768 0.85 CYP1A2 (0.41) GSK3BCYP1A2HSD17B10KMT2AGRIN2D
SCHEMBL7741417 0.85 CA12 (0.39) CYP1A2PRKAG1PRKAA1PRKAB1
SCHEMBL7741254 0.85 PTGES (0.37) PRKAG1PRKAA1PRKAB1KMT2AGRIN2D
SCHEMBL7742681 0.83 CDK5 (0.35) HSD17B10USP2KMT2AGRIN2DGRIN3B
SCHEMBL7740551 0.82 PRKAG1 (0.43) GSK3BCYP1A2PRKAG1PRKAA1PRKAB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420386-B1 SPINAL TRAUMATISM, EPILEPSY, CHRONIC NEURODEGENERATIVE DISEASES SUCH AS ALZHEIMER'S DISEASE, SCHIZOPHRENIA, LATERAL AMYOTROPHIC SCLEROSIS OR HUNTINGTON'S CHOREA. LES LABORATORIES SERVIER (FR) 2002-07-16 US disclosed