SCHEMBL7742768

SCHEMBL7742768

CCOP(=O)(OCC)c1cc2cc(-c3ccc([N+](=O)[O-])cc3)c(Cl)cc2[nH]c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
GSK3B P49841 1/20 0.41
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PGR P06401 1/20 0.37
NPBWR1 P48145 4/20 0.36
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7734964 0.89 ALDH1A1 (0.41) ALDH1A1MAPK1PGRGRIN2DGRIN3B
SCHEMBL7741117 0.86 PRKAG1 (0.37) CYP1A2GSK3BALDH1A1TSHRHSD17B10
SCHEMBL7739643 0.85 GSK3B (0.37) CYP1A2GSK3BALDH1A1TSHRHSD17B10
SCHEMBL7739842 0.85 PRKAG1 (0.42) CYP1A2ALDH1A1CYP3A4GRIN2DGRIN3B
SCHEMBL7740612 0.85 PRKAG1 (0.40) CYP1A2GSK3BALDH1A1CYP3A4GRIN2D
SCHEMBL7741417 0.84 CA12 (0.39) CYP1A2CA1CA2CYP3A4
SCHEMBL7741263 0.83 GRIA1 (0.41) CYP1A2GSK3BALDH1A1NPBWR1NPC1
SCHEMBL7740617 0.83 PTGES (0.36) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7741113 0.83 IDH1 (0.41) ALDH1A1PGRGRIN2DGRIN3BGRIN1
SCHEMBL6922992 0.82 GRIN2D (0.40) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420386-B1 SPINAL TRAUMATISM, EPILEPSY, CHRONIC NEURODEGENERATIVE DISEASES SUCH AS ALZHEIMER'S DISEASE, SCHIZOPHRENIA, LATERAL AMYOTROPHIC SCLEROSIS OR HUNTINGTON'S CHOREA. LES LABORATORIES SERVIER (FR) 2002-07-16 US disclosed