SCHEMBL7740425

SCHEMBL7740425

O=[N+]([O-])c1ccc(-n2cccc2)c(CO)c1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.47
MAPT P10636 3/20 0.44
NPSR1 Q6W5P4 2/20 0.44
HTT P42858 1/20 0.44
POLB P06746 2/20 0.43
ATM Q13315 1/20 0.43
ALDH1A1 P00352 3/20 0.42
LMNA P02545 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TSHR P16473 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
CTSB P07858 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740479 0.84 TDP1 (0.44) TDP1MAPTNPSR1HTTPOLB
SCHEMBL27495191 0.81 TDP1 (0.48) TDP1MAPTNPSR1HTTPOLB
SCHEMBL6562050 0.79 GPR35 (0.53) TDP1MAPTNPSR1HTTALDH1A1
SCHEMBL10914504 0.78 LMNA (0.64) TDP1MAPTNPSR1HTTALDH1A1
SCHEMBL7886140 0.77 TLR2 (0.45) MAPTHTTPOLBATMALDH1A1
SCHEMBL16824876 0.77 ALDH1A1 (0.67) MAPTNPSR1HTTPOLBALDH1A1
SCHEMBL6677996 0.77 GAA (0.57) TDP1MAPTNPSR1HTTALDH1A1
SCHEMBL2625708 0.76 TLR2 (0.47) MAPTHTTPOLBALDH1A1LMNA
SCHEMBL260788 0.76 CYP1A2 (0.51) TDP1MAPTPOLBATMALDH1A1
SCHEMBL29367937 0.76 CYP1A2 (0.51) TDP1MAPTPOLBATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed