SCHEMBL7740423

SCHEMBL7740423

Cc1c([N+](=O)[O-])cc(Br)c(-n2cccn2)c1CNC(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.37
MEN1 O00255 8/20 0.37
KMT2A Q03164 8/20 0.37
MAPT P10636 7/20 0.37
LMNA P02545 5/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
BRD4 O60885 2/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
HTT P42858 1/20 0.33
MDM2 Q00987 1/20 0.33
KDM4A O75164 1/20 0.32
PCSK9 Q8NBP7 1/20 0.32
KLKB1 P03952 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27513872 0.79 ALDH1A1 (0.38) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL7740445 0.78 MEN1 (0.39) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL7880092 0.69 EPAS1 (0.40) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL7872397 0.67 EPAS1 (0.35) MEN1KMT2AMAPTLMNARAB9A
SCHEMBL19717777 0.67 POLB (0.49) ALDH1A1MAPTLMNARAB9ANPSR1
SCHEMBL4404243 0.66 LMNA (0.54) LMNABRD4L3MBTL1KLKB1
SCHEMBL7738995 0.66 JAK2 (0.35) LMNABRD4CA12CA1CA2
SCHEMBL7738864 0.65 SYK (0.35) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL7740426 0.64 PDK1 (0.40) BRD4CA12CA1CA2CA9
SCHEMBL23118891 0.64 KLKB1 (0.40) ALDH1A1MEN1KMT2AMAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed