SCHEMBL7740641

SCHEMBL7740641

Cc1cc(Cl)cc(-c2[nH]c(C(F)(F)F)nc2-c2ccccc2S(C)(=O)=O)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.42
KMT2A Q03164 2/20 0.40
RAB9A P51151 2/20 0.40
ALOX5 P09917 1/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
BRAF P15056 1/20 0.36
PDE2A O00408 1/20 0.36
HSD11B1 P28845 3/20 0.36
P2RX7 Q99572 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
SDHB P21912 1/20 0.34
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089382 0.81 PTGS2 (0.54) PTGS2ESR1ESR2
SCHEMBL8802006 0.78 ALOX5 (0.42) PTGS2KMT2AALOX5MEN1POLB
SCHEMBL8810671 0.78 ALOX5 (0.46) PTGS2KMT2AALOX5MEN1POLB
SCHEMBL6735914 0.77 BRAF (0.38) PTGS2ESR1ESR2BRAF
SCHEMBL8814347 0.77 ALOX5 (0.40) PTGS2KMT2AALOX5MEN1POLB
SCHEMBL9079514 0.76 PTGS2 (0.43) PTGS2KMT2AALOX5MEN1POLB
SCHEMBL6738959 0.76 NR1H2 (0.35) PTGS2ALOX5ESR1ESR2BRAF
SCHEMBL6733161 0.75 NR1H2 (0.40) PTGS2KMT2ARAB9AESR1ESR2
SCHEMBL6723894 0.75 ESR1 (0.40) PTGS2ESR1ESR2BRAF
SCHEMBL6734567 0.74 SDHB (0.42) PTGS2RAB9AALOX5ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6426360-B1 ANTIARTHRITIC AGENTS G D SEARLE & CO. 2002-07-30 US disclosed