SCHEMBL7741933

SCHEMBL7741933

NC(=O)Nc1cccc(-c2ccc([N+](=O)[O-])cc2)c1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
ALDH1A1 P00352 2/20 0.49
MYC P01106 1/20 0.49
MAX P61244 1/20 0.49
POLB P06746 2/20 0.44
MAPK1 P28482 1/20 0.44
NPC1 O15118 4/20 0.43
ERO1A Q96HE7 1/20 0.43
RAB9A P51151 2/20 0.43
MITF O75030 1/20 0.43
HDAC2 Q92769 1/20 0.42
MAPT P10636 3/20 0.41
AR P10275 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
CD40 P25942 1/20 0.41
CD40LG P29965 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7621243 0.87 ALDH1A1 (0.56) MEN1KMT2AALDH1A1MYCMAX
SCHEMBL7611513 0.81 SLC6A3 (0.42) MEN1KMT2AALDH1A1POLBNPC1
SCHEMBL9754422 0.77 CA1 (0.48) ALDH1A1MYCMAXPOLBMAPK1
SCHEMBL17796945 0.77 ALDH1A1 (0.59) MEN1KMT2AALDH1A1MYCMAX
SCHEMBL17289272 0.77 ALDH1A1 (0.59) MEN1KMT2AALDH1A1MYCMAX
SCHEMBL7616828 0.77 IKBKB (0.52) MEN1KMT2AALDH1A1POLBNPC1
SCHEMBL16879409 0.74 ALDH1A1 (0.66) MEN1KMT2AALDH1A1MYCMAX
Phenylurea SCHEMBL27473020 0.74 MEN1 (0.63) MEN1KMT2AALDH1A1POLBMAPK1
SCHEMBL11612279 0.73 ALDH1A1 (0.54) MEN1KMT2AALDH1A1MYCMAX
SCHEMBL7615106 0.73 KIF11 (0.63) ALDH1A1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6417393-B1 TREATMENT OF SICKLE-CELL ANEMIA, BRAIN EDEMA FROM TUMORS OR ISCHEMIA, DIARRHEA, AND GLAUCOMA; HYPOTENSIVE, WOUND HEALING, ANTIINFLAMMATORY AND ANTIALLERGEN AGENTS NEUROSEARCH A/S (DK) 2002-07-09 US disclosed
EP-0906273-A1 PHENYL DERIVATIVES CONTAINING AN ACIDIC GROUP, THEIR PREPARATION AND THEIR USE AS CHLORIDE CHANNEL BLOCKERS NEUROSEARCH A/S (DK) 1999-04-07 EP disclosed
WO-1997045400-A1 PHENYL DERIVATIVES CONTAINING AN ACIDIC GROUP, THEIR PREPARATION AND THEIR USE AS CHLORIDE CHANNEL BLOCKERS NEUROSEARCH A/S (DK) 1997-12-04 WO disclosed