SCHEMBL7743876

SCHEMBL7743876

C[C@H](Cc1ccccc1)[C@@]1(n2cnc3c(N)ncnc32)O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.46
ADORA3 P0DMS8 5/20 0.46
ADORA2B P29275 2/20 0.46
ADORA1 P30542 2/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46
TSHR P16473 1/20 0.46
ALOX12 P18054 1/20 0.46
NFKB1 P19838 1/20 0.46
HIF1A Q16665 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
PMP22 Q01453 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
PI4KA P42356 2/20 0.43
PI4K2B Q8TCG2 2/20 0.43
PI4K2A Q9BTU6 2/20 0.43
PI4KB Q9UBF8 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL859642 1.00 ADORA2A (0.46) ADORA2AADORA3ADORA2BADORA1TP53
Benzene SCHEMBL27650186 0.87 PI4KA (0.48) ADORA2AADORA3ADORA2BADORA1PI4KA
SCHEMBL13269091 0.87 PI4KA (0.45) ADORA2AADORA3ADORA2BADORA1PI4KA
SCHEMBL5525776 0.87 PI4KA (0.45) ADORA2AADORA3ADORA2BADORA1PI4KA
SCHEMBL13268818 0.87 PI4KA (0.45) ADORA2AADORA3ADORA2BADORA1PI4KA
SCHEMBL6829143 0.86 PI4KA (0.48) ADORA2AADORA3ADORA2BADORA1HIF1A
SCHEMBL29721329 0.85 ADORA3 (0.50) ADORA2AADORA3ADORA2BADORA1PI4KA
SCHEMBL7435441 0.85 ADORA3 (0.50) ADORA2AADORA3ADORA2BADORA1PI4KA
SCHEMBL10710442 0.85 ADORA3 (0.46) ADORA2AADORA3ADORA2BADORA1PI4KA
SCHEMBL2270700 0.84 ADORA2A (0.51) ADORA2AADORA3ADORA2BADORA1PI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708781-B1 A 3 ADENOSINE RECEPTOR AGONISTS USA (US) 2001-10-04 EP disclosed
EP-0708781-A1 A 3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, Department of Health and Human Services (US) 1996-05-01 EP disclosed
WO-1995002604-A1 A3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-01-26 WO disclosed