Lithium Ion

Lithium Ion

SCHEMBL7743896

N#Cc1ccc(CC(C(=O)[O-])c2cnc[nH]2)cc1F.[Li+]

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Lithium Ion. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CPB2 Q96IY4 11/20 0.50
CPA1 P15085 1/20 0.44
CPB1 P15086 3/20 0.42
DAO P14920 2/20 0.40
CYP11B2 P19099 4/20 0.38
CYP11B1 P15538 3/20 0.38
CYP19A1 P11511 1/20 0.36
CACNA1H O95180 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7743898 0.88 CPB2 (0.62) CPB2CPA1CPB1DAOCYP19A1
SCHEMBL7743300 0.85 CPB2 (0.48) CPB2CPA1CPB1DAOCYP11B2
SCHEMBL7704747 0.75 CACNA1H (0.40) CPB2DAOCYP11B2CYP11B1CYP19A1
SCHEMBL7053727 0.69 CPA1 (0.71) CPB2CPA1CPB1CYP19A1
Hydrochloric Acid SCHEMBL8495732 0.69 CPA1 (0.69) CPB2CPA1CPB1CYP19A1
SCHEMBL7704752 0.67 DAO (0.40) DAOCYP11B2CYP11B1CACNA1H
SCHEMBL8865742 0.67 CPA1 (0.76) CPB2CPA1CPB1CYP19A1
SCHEMBL25220822 0.67 TRPV4 (0.45) DAOCYP11B2CYP11B1CACNA1H
SCHEMBL2722813 0.66 TRPV4 (0.47) DAOCYP11B2CYP11B1CACNA1H
SCHEMBL7086614 0.66 CPA1 (0.51) CPB2CPA1CPB1CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091736-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2001-10-24 EP disclosed
EP-1091736-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2001-04-18 EP disclosed
WO-2000001382-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-01-13 WO disclosed